API Intermediates

Structure Intermediate Name CAS No API/ END USE
Ethyl 3-(3-amino-4-(methyl amino)-N-(pyridin-2-yl) benzamido) propanoate/ DGT-3 212322-56-0 Dabigatran
2-(4-Cyanophenylamino) Acetic Acid/ DGT-4 42288-26-6 Dabigatran
Ethyl-3-[[[2-[[(4-cyanophenyl) amino] methyl]-1methyl-1H-benzimidazol-5-yl] carbonyl] pyridine-2-ylamino] propionate/DGT5 211915-84-3 Dabigatran
Ethyl 3-(2-(((4-carbamimidoylphenyl)amino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate hydrochloride//DGT6 211914-50-0 Dabigatran
2,3,4,6-tetrakis-o-trimethylsilyl-d-gluconolactone/ DGL1 32384-65-9 Dapagliflozin/ Empa Canagliflozin
4-Chloro Benzhydryl Piperazine/ CBP3 303-26-4 Cetirizine / Buclizine/ Meclizine/Hydroxyzine/ Etodroxizine
Formamidine acetate salt / ACF 3473-63-0 Itraconazole/ Ibrutinib/Tofacitinib
5-chloro-4-amino-2,1,3-benzothiadiazole / ABT3 30536-19-7 Tizanidine
N N’ Di isopropyl carbodiimide// NNDIC 693-13-0 Tirzepatide// Liraglutide/Semaglutide
8-Chloro-5,10-dihydro-11H-dibenzo[b,e][1,4]-diazepin-11-one, /COD-3 50892-62-1 Clozapine
2-(2-Aminothiazol-4-yl) acetic acid / AAA-2 29676-71-9 Mirabegron
2-(4-nitrophenyl)ethanamine hydrochloride /NPA-2 29968-78-3 Mirabegron
(R)-2-Hydroxy-N-(4-nitrophenethyl)-2-phenylacetamide/MGN-1 521284-19-5 Mirabegron
(R)-2-(4-nitrophenethylamino)-1- Phenylethanol MGN 2 223673-34-5 Mirabegron
(R)-2-(4-nitrophenethylamino)-1-phenylethanol hydrochloride/ MGN 2HCL 521284-21-9 Mirabegron
(R)-2-((4-Aminophenethyl)amino)-1-phenylethanol//MGN3Base 391901-45-4 Mirabegron
(R)-2-(4-aminophenethylamino)-1-Phenylethanol hydrochloride/ MGN 3// N-1 521284-22-0 Mirabegron
Methyl 5-tert-butyl-2-hydroxy benzoate//SAS-2 52888-72-9 Deutivacaftor
2-Butyl-1,3-diazaspiro[4.4]non-1-en-4-oneHydrochloride/Spiro Compound/TBI-3 151257-01-1 Irbesartan
(betaR,gammaR)-gamma-Ethyl-3-methoxy-N,N,beta-trimethylbenzenepropanamine hydrochloride(N-1) 175591-17-0 Tapentadol
(2-ethoxyethyl 4-methylbenzenesulfonate)// EPB-1 17178-11-9 Bilastine
2-(Piperidin-4 yl)-1H- Benzo[d]imidazole//EPB2 38385-95-4 Bilastine
1-(2-Ethoxyethyl)-2-(piperidin-4-yl)-1H-benzo[d]imidazole hydrochloride//EPB4 1841081-72-8 Bilastine
Methyl 2-(4-(2-chloroethyl) phenyl)-2-Methyl propanoate//CPM-3 1181267-33-3 Bilastine
N,N-Dimethylamino propiophenone hydrochloride /AMT1 879-72-1 Fluoxetine
N,N-Dimethyl-3-phenyl-3-chloropropylamine hydrochloride/ AMT2 1011-59-2 Atomoxetine
N,N-dimethyl-3-phenyl-3-(O-tolyloxy)propan-1-amine oxalate/ AMT3 107688-86-8 Atomoxetine
tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate 571188-59-5 Ribociclib
1-(4-Morpholinophenyl)guanidine//MAN-3 247234-41-9 Momelotinib
4-((tert-butoxycarbonyl)amino)piperidine-4-carboxylic acid//CPS- 252720-31-3 Capivasertib
1-(Cyclopropylcarbonyl) piperazine hydrochloride/CPP 1021298-67-8 Olaparib
Dimethyl (3-oxo-1,3-dihydroisobenzofuran-1-yl)phosphonate/OLP1 61260-15-9 Olaparib
4-(Piperidin-4yl) morpholine hydrochloride /PPD2Hcl 550370-31-5 Alectinib
4-(Piperidin-4yl) morpholine//PPD2 53617-35-9 Alectinib
2-Bromo-4-Nitro Imidazole/ BNI-2 65902-59-2 Delamanid/Pretomanid
(R)-2-(tert-butoxycarbonylamino)-2-phenylethyl methanesulfonate//IEL 102089-75-8 Elagolix
9,10-dimethoxy-2-(2,4,6-trimethylanilino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one//ETS4 76536-66-8 Ensifentrine
N-Methoxy-N-methylacetamide) NMMA, 78191-00-1 Pyridine Derivatives
2-(Chloromethyl)-4-methylquinazoline/ CLM-1 109113-72-6 Linagliptin/ Trelagliptin/ Alogliptin
8-Bromo-7-(2-butyn-1-yl)-3-methylxanthine BMP-2 666816-98-4 Linagliptin/ Trelagliptin/ Alogliptin
1,4,7-Trimethyl-1,4,7-Triazacyclononane/ TTC2 (Stabilised with sodium bi carbonate) 96556-05-7 Speciality chemical used in tanning/ detergents and as additive
(-)-4-Chlorobenzhydrylamine/LCH2 163837-57-8 Levocetirizine
N,N-bis(2-Chloroethyl)-4-MethylbenzeneSulfonamide/CMS 42137-88-2 Levocetirizine
Under Development
(R)- N-methyl-3-phenyl-3-(O-tolyloxy)propan-1-amine (s)- (+)- Mandelate //(R)-tomoxetine (S)-(+)- mandelic acid salt /RTM-4 83113-55-7 Atomoxetine
Ethyl 3-amino-1H-pyrazole 4-carboxylate //EPC 6994-25-8 Allopurinol
2,4-Dichloro-7h-Pyrrolo2,3-Dpyrimidine 90123-66-4 Tofacitinib
4-Amino-2,6-dichlorophenol / DNP-1 5930-28-9 Resmetirom
6-(4-amino-2,6-dichlorophenoxy)-4-isopropylpyridazin-3(2H)-one// RCM-4 920509-28-0 Resmetirom
(S)-tert-butyl (1-aMino-3-(4-iodophenyl)-1-oxopropan-2-yl)carbamate//BCB3 868694-44-4 Brensocatib
3-(Hexyloxy)-4-(pyridin-3-yl)-1,2,5-thiadiazole 131987-69-4 Xanomeline
5-Methyl-1,3,4-oxadiazole-2-carboxylic acid potassium salt.// PMC-3 888504-28-7 Raltegravir
1-((iso cyano methyl)sulfonyl)-4-methylbenzene// TosMIC 36635-61-7 Bempedoic Acid
3-Aminopiperidine-2,6-dione hydrochloride,/DPA3 24666-56-6 Lenalidomide
Methyl-2-bromomethyl-3-nitrobenzoate/NBM2 98475-07-1 Lenalidomide
4-Bromo-1-chloro-2-[(4-ethoxyphenyl)methyl]benzene//DGP2 461432-23-5 Dapagliflozin
4-Morpholineacetic acid hydrochloride/CAR 89531-58-8 Carfilzomib
6-Chloro-3-(1-Methylethyl)-2,4-(1h,3h)-Pyrimidinedione 887581-47-7 Mavacamten
1-isopropylpyrimidine-2,4,6(1H,3H,5H)-trione 69998-14-7 Mavacamten
(S)-3-((2R,5S)-5-(4-Fluorophenyl)-2-((S)-((4-fluorophenyl)amino)(4-((trimethylsilyl)oxy)phenyl)methyl)-5-((trimethylsilyl)oxy)pentanoyl)-4-phenyloxazolidin-2-one 272778-12-8 Ezetimibe
4-Octylphenyl Ethanol//FNG2A 162358-05-6 Fingolimod
3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-ol 1779428-05-5 Acoramidis
4-(3-bromopropyl)-3,5-dimethyl-1H-pyrazole 2167368-32-1 Acoramidis
3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazine-6-carboxylic acid 134997-87-8 Balcinaranone
N-Boc-Piperidine-4-carboxylic acid methyl ester 124443-68-1 Muvalaplin
1-tert-butyl 4-methyl 4-(3-bromobenzyl)piperidine-1,4-dicarboxylate 3086955-18-9 Muvalaplin
4-[(3-bromophenyl)methyl]-1,4-Piperidinedicarboxylic acid 1-(1,1-dimethylethyl)ester 1187172-25-3 Muvalaplin
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