| Structure | Intermediate Name | CAS No | API/ END USE |
|---|---|---|---|
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2-(2-Aminothiazol-4-yl) acetic acid / AAA-2 | 29676-71-9 | Mirabegron |
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2-(4-nitrophenyl)ethanamine hydrochloride /NPA-1 | 29968-78-3 | Mirabegron |
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(R)-2-Hydroxy-N-(4-nitrophenethyl)-2-phenylacetamide/MGN-1 | 521284-19-5 | Mirabegron |
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(R)-2-(4-nitrophenethylamino)-1- Phenylethanol MGN 2Base | 223673-34-5 | Mirabegron |
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(R)-2-(4-nitrophenethylamino)-1-phenylethanol hydrochloride/ MGN 2HCL | 521284-21-9 | Mirabegron |
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(R)-2-((4-Aminophenethyl)amino)-1-phenylethanol//MGN3Base | 391901-45-4 | Mirabegron |
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(R)-2-(4-aminophenethylamino)-1-Phenylethanol hydrochloride/ MGN 3// N-1 | 521284-22-0 | Mirabegron |
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4-Chloro Benzhydryl Piperazine/ CBP-3 | 303-26-4 | Cetirizine / Buclizine/ Meclizine/Hydroxyzine/ Etodroxizine |
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N N’ Di isopropyl carbodiimide// DIC-1 | 693-13-0 | Tirzepatide// Liraglutide/Semaglutide |
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5-chloro-4-amino-2,1,3-benzothiadiazole / ABT-3 | 30536-19-7 | Tizanidine |
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N,N-dichloroethyl-4-methoxy benzene sulphonamide / MBS-2 | 86357-59-7 | Levocetirizine |
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8-Chloro-5,10-dihydro-11H-dibenzo[b,e][1,4]-diazepin-11-one, /CODD-3 | 50892-62-1 | Clozapine |
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4-((tert-butoxycarbonyl)amino)piperidine-4-carboxylic acid//CPS-4 | 252720-31-3 | Capivasertib |
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1-(4-Morpholinophenyl)guanidine//MAN-3 | 247234-41-9 | Momelotinib |
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N-Methoxy-N-methylacetamide) NMMA, | 78191-00-1 | Alpelisib |
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(betaR,gammaR)-gamma-Ethyl-3-methoxy-N,N,beta-trimethylbenzenepropanamine hydrochloride(N-1) | 175591-17-0 | Tapentadol |
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Formamidine acetate salt / ACF | 3473-63-0 | Itraconazole/ Ibrutinib/Tofacitinib |
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Ethyl 3-amino-1H-pyrazole 4-carboxylate //EPC | 6994-25-8 | Allopurinol |
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Methyl 5-tert-butyl-2-hydroxy benzoate//SAS-2 | 52888-72-9 | Deutivacaftor |
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Tert-butyl 2,6-dichloronicotinate// TDC-1 | 1013647-75-0 | Elexacaftor |
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4-oxo-1, 4-dihydroquinoline-3-carboxylic acid // ACQ-3P |
13721-01-2 | Ivacaftor |
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5-Amino-2,4-ditert-butylphenol//DTB-3 | 873055-58-4 | Ivacaftor |
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2,3,4,6-tetrakis-o-trimethylsilyl-d-gluconolactone/ DGL-1 | 32384-65-9 | Dapagliflozin/ Empagliflozin Canagliflozin |
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2-Butyl-1,3-diazaspiro[4.4]non-1-en-4-oneHydrochloride/Spiro Compound/TBI-3 | 151257-01-1 | Irbesartan |
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N,N-Dimethylamino propiophenone hydrochloride /AMT-1 | 879-72-1 | Fluoxetine |
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N,N-Dimethyl-3-phenyl-3-chloropropylamine hydrochloride/ AMT-2 | 1011-59-2 | Atomoxetine |
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N,N-dimethyl-3-phenyl-3-(O-tolyloxy)propan-1-amine oxalate/ AMT-3 | 107688-86-8 | Atomoxetine |
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2-Bromo-4-Nitro Imidazole/ BNI-2 | 65902-59-2 | Delamanid/Pretomanid |
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tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate - RBC-2 | 571188-59-5 | Ribociclib/ Palbociclib |
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1-(Cyclopropylcarbonyl) piperazine hydrochloride/CPPHCL | 1021298-67-8 | Olaparib |
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Dimethyl (3-oxo-1,3-dihydroisobenzofuran-1-yl)phosphonate/OLP1 | 61260-15-9 | Olaparib |
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4-(Piperidin-4yl) morpholine hydrochloride /PPD2Hcl | 550370-31-5 | Alectinib |
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4-(Piperidin-4yl) morpholine//PPD2 | 53617-35-9 | Alectinib |
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2-(4-ethyl-3-iodophenyl)-2-Methylpropanoic acid//EIP-4 | 1256584-73-2 | Alectinib |
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Tert-butyl 6-cyano-2-(2-(4-ethyl-3-iodophenyl)propan-2-yl)-1H-indole-3- carboxylate//TCC-3 | 1256584-75-4 | Alectinib |
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4-Morpholineacetic acid hydrochloride/CAR-1 | 89531-58-8 | Carfilzomib |
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4-Amino-2,6-dichlorophenol / DAP-2 | 5930-28-9 | Resmetirom |
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3,6-dichloro-4-isopropyl pyridazine / RMT-3 | 107228-51-3 | Resmetirom |
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3,5-dichloro-4-((6-chloro-4-isopropyl pyridazin-3-yl) oxy) aniline / RMT-4 | 920509-27-9 | Resmetirom |
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6-(4-amino-2,6-dichlorophenoxy)-4-isopropylpyridazin-3(2H)-one// RMC-5 | 920509-28-0 | Resmetirom |
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N-Cyano acetyl urethane //NCU | 6629-04-5 | Resmetirom |
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(S)-tert-butyl (1-aMino-3-(4-iodophenyl)-1-oxopropan-2-yl)carbamate//BCB3 | 868694-44-4 | Brensocatib |
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3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2(3H)- benzoxazolone//MTB-3 | 1220696-32-1 | Brensocatib |
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5-Chloro-3-methyl-2(3H)-benzoxazolone / COZ-2 | 5790-90-9 | Brensocatib |
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5-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-3-methylbenzo[d]oxazol-2(3H)-one//COZ-3 | 1802149-87-6 | Brensocatib |
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9,10-dimethoxy-2-(2,4,6-trimethylanilino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one//ETS-4 | 76536-66-8 | Ensifentrine |
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3-Chloro-4-(Pyridin-3-yl)-1, 2, 5-Thiadiazole / HPT-2 | 131986-28-2 | Xanomeline |
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3-(Hexyloxy)-4-(pyridin-3-yl)-1,2,5-thiadiazole / HPT-3 | 131987-69-4 | Xanomeline |
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(+)-2,3-O-Isopropylidene-L-threitol//TRS-3 | 50622-09-8 | Treosulfan |
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(R)-2-(tert-butoxycarbonylamino)-2-phenylethyl methanesulfonate//IEL | 102089-75-8 | Elagolix |
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3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-ol | 1779428-05-5 | Acoramidis |
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N-Boc-O-methyl-L-tyrosine / LTC-2 | 53267-93-9 | Carbetocin |
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Ethyl 3-(3-amino-4-(methyl amino)-N-(pyridin-2-yl) benzamido) propanoate/ DGT-3 | 212322-56-0 | Dabigatran |
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2-(4-Cyanophenylamino) Acetic Acid/ DGT-4 | 42288-26-6 | Dabigatran |
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Ethyl-3-[[[2-[[(4-cyanophenyl) amino] methyl]-1methyl-1H-benzimidazol-5-yl] carbonyl] pyridine-2-ylamino] propionate/DGT5 | 211915-84-3 | Dabigatran |
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Ethyl 3-(2-(((4-carbamimidoylphenyl)amino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate hydrochloride//DGT6 | 211914-50-0 | Dabigatran |
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(2-ethoxyethyl 4-methylbenzenesulfonate)// EPB-1 | 17178-11-9 | Bilastine |
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2-(Piperidin-4 yl)-1H- Benzo[d]imidazole//EPB2 | 38385-95-4 | Bilastine |
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1-(2-Ethoxyethyl)-2-(piperidin-4-yl)-1H-benzo[d]imidazole hydrochloride//BST-4 | 1841081-72-8 | Bilastine |
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Methyl 2-(4-(2-chloroethyl) phenyl)-2-Methyl propanoate//CPM-3 | 1181267-33-3 | Bilastine |
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2-(Chloromethyl)-4-methylquinazoline/ CLM-1 | 109113-72-6 | Linagliptin/ Trelagliptin/ Alogliptin |
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8-Bromo-7-(2-butyn-1-yl)-3-methylxanthine BMP-2 | 666816-98-4 | Linagliptin/ Trelagliptin/ Alogliptin |
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1-tert-Butyl-3-ethylcarbodiimide // TEC-3 | 1433-27-8 | Peptide coupling Reagent |
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1,4,7-Trimethyl-1,4,7-Triazacyclononane/ TTC-4 (Stabilised with sodium bi carbonate) | 96556-05-7 | Speciality chemical used in tanning/ detergents and as additive |
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(-)-4-Chlorobenzhydrylamine/LCH2 | 163837-57-8 | Levocetirizine |
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N,N-bis(2-Chloroethyl)-4-MethylbenzeneSulfonamide/CMS | 42137-88-2 | Levocetirizine |
| Under Development | |||
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2-Butynoic Acid //BYA-3 | 590-93-2 | Acalabrutinib |
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(R)- N-methyl-3-phenyl-3-(O-tolyloxy)propan-1-amine (s)- (+)- Mandelate //(R)-tomoxetine (S)-(+)- mandelic acid salt /RTM-4 | 83113-55-7 | Atomoxetine |
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Methyl 4-Fluoro-3-Hydroxybenzoate / ACM-1 | 214822-96-5 | Acoramidis |
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Benzoic acid, 3-[3-(3,5-dimethyl-1H-pyrazol-4-yl) propoxy]-4-fluoro-, methyl ester | 1446701-54-7 | Acoramidis |
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2-Amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide | 302964-24-5 | Dasatinib |
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4,6-dichloro-2-methylpyrimidine | 1780-26-3 | Dasatinib |
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4-Bromo-1-chloro-2-[(4-ethoxyphenyl)methyl]benzene//DGP2 | 461432-23-5 | Dapagliflozin |
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(S)-3-((2R,5S)-5-(4-Fluorophenyl)-2-((S)-((4-fluorophenyl)amino)(4-((trimethylsilyl)oxy)phenyl)methyl)-5-((trimethylsilyl)oxy)pentanoyl)-4-phenyloxazolidin-2-one | 272778-12-8 | Ezetimibe |
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4-Octylphenyl Ethanol//FNG2A | 162358-05-6 | Fingolimod |
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N,O-Dibenzylated formoterol//NDF | 43229-70-5 | Formoterol Fumarate |
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N,N-Dimethylpiperidin-4-amine Dihydrochloride | 4876-59-9 | Gedatolisib |
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2,4-Diamino-6-(4-nitrophenyl)-1,3,5-triazine | 29366-73-2 | Gedatolisib |
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1,3,5-Triazine, 2,4-di-4-morpholinyl-6-(4-nitrophenyl)- | 2161412-22-0 | Gedatolisib |
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4-(4,6-dimorpholino-1,3,5-triazin-2-yl)aniline | 1197159-91-3 | Gedatolisib |
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(4-Aminophenyl)(4-(dimethylamino)piperidin-1-yl)methanone | 1605251-03-3 | Gedatolisib |
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3-Aminopiperidine-2,6-dione hydrochloride,/DPA3 | 24666-56-6 | Lenalidomide |
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Methyl-2-bromomethyl-3-nitrobenzoate/NBM2 | 98475-07-1 | Lenalidomide |
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6-Chloro-3-(1-Methylethyl)-2,4-(1h,3h)-Pyrimidinedione | 887581-47-7 | Mavacamten |
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1-isopropylpyrimidine-2,4,6(1H,3H,5H)-trione | 69998-14-7 | Mavacamten |
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5-chloro-2-(piperidin-4-yl)pyrimidine hydrochloride | 1402666-88-9 | Nerandomilast |
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5-Methyl-1,3,4-oxadiazole-2-carboxylic acid potassium salt.// PMC-3 | 888504-28-7 | Raltegravir |
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4-chloro-7H-pyrrolo [2,3-d]pyrimidine// TFN-3 | 3680-69-1 | Tofacitinib,Barcitinib Ruxolitinib |
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(R)-5-Cyclopentylpyrazolidin-3-one D(-)-Tartaric acid// CPD-5 | 2102675-37-4 | Ruxolitinib |