API Intermediates

Structure Intermediate Name CAS No API/ END USE
2-(2-Aminothiazol-4-yl) acetic acid / AAA-2 29676-71-9 Mirabegron
2-(4-nitrophenyl)ethanamine hydrochloride /NPA-1 29968-78-3 Mirabegron
(R)-2-Hydroxy-N-(4-nitrophenethyl)-2-phenylacetamide/MGN-1 521284-19-5 Mirabegron
(R)-2-(4-nitrophenethylamino)-1- Phenylethanol MGN 2Base 223673-34-5 Mirabegron
(R)-2-(4-nitrophenethylamino)-1-phenylethanol hydrochloride/ MGN 2HCL 521284-21-9 Mirabegron
(R)-2-((4-Aminophenethyl)amino)-1-phenylethanol//MGN3Base 391901-45-4 Mirabegron
(R)-2-(4-aminophenethylamino)-1-Phenylethanol hydrochloride/ MGN 3// N-1 521284-22-0 Mirabegron
4-Chloro Benzhydryl Piperazine/ CBP-3 303-26-4 Cetirizine / Buclizine/ Meclizine/Hydroxyzine/ Etodroxizine
N N’ Di isopropyl carbodiimide// DIC-1 693-13-0 Tirzepatide// Liraglutide/Semaglutide
5-chloro-4-amino-2,1,3-benzothiadiazole / ABT-3 30536-19-7 Tizanidine
N,N-dichloroethyl-4-methoxy benzene sulphonamide / MBS-2 86357-59-7 Levocetirizine
8-Chloro-5,10-dihydro-11H-dibenzo[b,e][1,4]-diazepin-11-one, /CODD-3 50892-62-1 Clozapine
4-((tert-butoxycarbonyl)amino)piperidine-4-carboxylic acid//CPS-4 252720-31-3 Capivasertib
1-(4-Morpholinophenyl)guanidine//MAN-3 247234-41-9 Momelotinib
N-Methoxy-N-methylacetamide) NMMA, 78191-00-1 Alpelisib
(betaR,gammaR)-gamma-Ethyl-3-methoxy-N,N,beta-trimethylbenzenepropanamine hydrochloride(N-1) 175591-17-0 Tapentadol
Formamidine acetate salt / ACF 3473-63-0 Itraconazole/ Ibrutinib/Tofacitinib
Ethyl 3-amino-1H-pyrazole 4-carboxylate //EPC 6994-25-8 Allopurinol
Methyl 5-tert-butyl-2-hydroxy benzoate//SAS-2 52888-72-9 Deutivacaftor
Tert-butyl 2,6-dichloronicotinate// TDC-1 1013647-75-0 Elexacaftor
4-oxo-1, 4-dihydroquinoline-3-carboxylic acid //
ACQ-3P
13721-01-2 Ivacaftor
5-Amino-2,4-ditert-butylphenol//DTB-3 873055-58-4 Ivacaftor
2,3,4,6-tetrakis-o-trimethylsilyl-d-gluconolactone/ DGL-1 32384-65-9 Dapagliflozin/ Empagliflozin Canagliflozin
2-Butyl-1,3-diazaspiro[4.4]non-1-en-4-oneHydrochloride/Spiro Compound/TBI-3 151257-01-1 Irbesartan
N,N-Dimethylamino propiophenone hydrochloride /AMT-1 879-72-1 Fluoxetine
N,N-Dimethyl-3-phenyl-3-chloropropylamine hydrochloride/ AMT-2 1011-59-2 Atomoxetine
N,N-dimethyl-3-phenyl-3-(O-tolyloxy)propan-1-amine oxalate/ AMT-3 107688-86-8 Atomoxetine
2-Bromo-4-Nitro Imidazole/ BNI-2 65902-59-2 Delamanid/Pretomanid
tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate - RBC-2 571188-59-5 Ribociclib/ Palbociclib
1-(Cyclopropylcarbonyl) piperazine hydrochloride/CPPHCL 1021298-67-8 Olaparib
Dimethyl (3-oxo-1,3-dihydroisobenzofuran-1-yl)phosphonate/OLP1 61260-15-9 Olaparib
4-(Piperidin-4yl) morpholine hydrochloride /PPD2Hcl 550370-31-5 Alectinib
4-(Piperidin-4yl) morpholine//PPD2 53617-35-9 Alectinib
2-(4-ethyl-3-iodophenyl)-2-Methylpropanoic acid//EIP-4 1256584-73-2 Alectinib
Tert-butyl 6-cyano-2-(2-(4-ethyl-3-iodophenyl)propan-2-yl)-1H-indole-3- carboxylate//TCC-3 1256584-75-4 Alectinib
4-Morpholineacetic acid hydrochloride/CAR-1 89531-58-8 Carfilzomib
4-Amino-2,6-dichlorophenol / DAP-2 5930-28-9 Resmetirom
3,6-dichloro-4-isopropyl pyridazine / RMT-3 107228-51-3 Resmetirom
3,5-dichloro-4-((6-chloro-4-isopropyl pyridazin-3-yl) oxy) aniline / RMT-4 920509-27-9 Resmetirom
6-(4-amino-2,6-dichlorophenoxy)-4-isopropylpyridazin-3(2H)-one// RMC-5 920509-28-0 Resmetirom
N-Cyano acetyl urethane //NCU 6629-04-5 Resmetirom
(S)-tert-butyl (1-aMino-3-(4-iodophenyl)-1-oxopropan-2-yl)carbamate//BCB3 868694-44-4 Brensocatib
3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2(3H)- benzoxazolone//MTB-3 1220696-32-1 Brensocatib
5-Chloro-3-methyl-2(3H)-benzoxazolone / COZ-2 5790-90-9 Brensocatib
5-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-3-methylbenzo[d]oxazol-2(3H)-one//COZ-3 1802149-87-6 Brensocatib
9,10-dimethoxy-2-(2,4,6-trimethylanilino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one//ETS-4 76536-66-8 Ensifentrine
3-Chloro-4-(Pyridin-3-yl)-1, 2, 5-Thiadiazole / HPT-2 131986-28-2 Xanomeline
3-(Hexyloxy)-4-(pyridin-3-yl)-1,2,5-thiadiazole / HPT-3 131987-69-4 Xanomeline
(+)-2,3-O-Isopropylidene-L-threitol//TRS-3 50622-09-8 Treosulfan
(R)-2-(tert-butoxycarbonylamino)-2-phenylethyl methanesulfonate//IEL 102089-75-8 Elagolix
3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-ol 1779428-05-5 Acoramidis
N-Boc-O-methyl-L-tyrosine / LTC-2 53267-93-9 Carbetocin
Ethyl 3-(3-amino-4-(methyl amino)-N-(pyridin-2-yl) benzamido) propanoate/ DGT-3 212322-56-0 Dabigatran
2-(4-Cyanophenylamino) Acetic Acid/ DGT-4 42288-26-6 Dabigatran
Ethyl-3-[[[2-[[(4-cyanophenyl) amino] methyl]-1methyl-1H-benzimidazol-5-yl] carbonyl] pyridine-2-ylamino] propionate/DGT5 211915-84-3 Dabigatran
Ethyl 3-(2-(((4-carbamimidoylphenyl)amino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate hydrochloride//DGT6 211914-50-0 Dabigatran
(2-ethoxyethyl 4-methylbenzenesulfonate)// EPB-1 17178-11-9 Bilastine
2-(Piperidin-4 yl)-1H- Benzo[d]imidazole//EPB2 38385-95-4 Bilastine
1-(2-Ethoxyethyl)-2-(piperidin-4-yl)-1H-benzo[d]imidazole hydrochloride//BST-4 1841081-72-8 Bilastine
Methyl 2-(4-(2-chloroethyl) phenyl)-2-Methyl propanoate//CPM-3 1181267-33-3 Bilastine
2-(Chloromethyl)-4-methylquinazoline/ CLM-1 109113-72-6 Linagliptin/ Trelagliptin/ Alogliptin
8-Bromo-7-(2-butyn-1-yl)-3-methylxanthine BMP-2 666816-98-4 Linagliptin/ Trelagliptin/ Alogliptin
1-tert-Butyl-3-ethylcarbodiimide // TEC-3 1433-27-8 Peptide coupling Reagent
1,4,7-Trimethyl-1,4,7-Triazacyclononane/ TTC-4 (Stabilised with sodium bi carbonate) 96556-05-7 Speciality chemical used in tanning/ detergents and as additive
(-)-4-Chlorobenzhydrylamine/LCH2 163837-57-8 Levocetirizine
N,N-bis(2-Chloroethyl)-4-MethylbenzeneSulfonamide/CMS 42137-88-2 Levocetirizine
Under Development
2-Butynoic Acid //BYA-3 590-93-2 Acalabrutinib
(R)- N-methyl-3-phenyl-3-(O-tolyloxy)propan-1-amine (s)- (+)- Mandelate //(R)-tomoxetine (S)-(+)- mandelic acid salt /RTM-4 83113-55-7 Atomoxetine
Methyl 4-Fluoro-3-Hydroxybenzoate / ACM-1 214822-96-5 Acoramidis
Benzoic acid, 3-[3-(3,5-dimethyl-1H-pyrazol-4-yl) propoxy]-4-fluoro-, methyl ester 1446701-54-7 Acoramidis
2-Amino-N-(2-chloro-6-methylphenyl)thiazole-5-carboxamide 302964-24-5 Dasatinib
4,6-dichloro-2-methylpyrimidine 1780-26-3 Dasatinib
4-Bromo-1-chloro-2-[(4-ethoxyphenyl)methyl]benzene//DGP2 461432-23-5 Dapagliflozin
(S)-3-((2R,5S)-5-(4-Fluorophenyl)-2-((S)-((4-fluorophenyl)amino)(4-((trimethylsilyl)oxy)phenyl)methyl)-5-((trimethylsilyl)oxy)pentanoyl)-4-phenyloxazolidin-2-one 272778-12-8 Ezetimibe
4-Octylphenyl Ethanol//FNG2A 162358-05-6 Fingolimod
N,O-Dibenzylated formoterol//NDF 43229-70-5 Formoterol Fumarate
N,N-Dimethylpiperidin-4-amine Dihydrochloride 4876-59-9 Gedatolisib
2,4-Diamino-6-(4-nitrophenyl)-1,3,5-triazine 29366-73-2 Gedatolisib
1,3,5-Triazine, 2,4-di-4-morpholinyl-6-(4-nitrophenyl)- 2161412-22-0 Gedatolisib
4-(4,6-dimorpholino-1,3,5-triazin-2-yl)aniline 1197159-91-3 Gedatolisib
(4-Aminophenyl)(4-(dimethylamino)piperidin-1-yl)methanone 1605251-03-3 Gedatolisib
3-Aminopiperidine-2,6-dione hydrochloride,/DPA3 24666-56-6 Lenalidomide
Methyl-2-bromomethyl-3-nitrobenzoate/NBM2 98475-07-1 Lenalidomide
6-Chloro-3-(1-Methylethyl)-2,4-(1h,3h)-Pyrimidinedione 887581-47-7 Mavacamten
1-isopropylpyrimidine-2,4,6(1H,3H,5H)-trione 69998-14-7 Mavacamten
5-chloro-2-(piperidin-4-yl)pyrimidine hydrochloride 1402666-88-9 Nerandomilast
5-Methyl-1,3,4-oxadiazole-2-carboxylic acid potassium salt.// PMC-3 888504-28-7 Raltegravir
4-chloro-7H-pyrrolo [2,3-d]pyrimidine// TFN-3 3680-69-1 Tofacitinib,Barcitinib Ruxolitinib
(R)-5-Cyclopentylpyrazolidin-3-one D(-)-Tartaric acid// CPD-5 2102675-37-4 Ruxolitinib
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